publicações selecionadas
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artigo académico
- 2-Aryladenine Derivatives as a Potent Scaffold for Adenosine Receptor Antagonists: The 6-Morpholino Derivatives. Biomolecules. 2024
- A Tandem Reaction in the Synthesis of New 4,8-Disubstituted-pyrimido[5,4-d]pyrimidine Derivatives. Asian Journal of Organic Chemistry. 2023
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artigo de revista
- Synthesis of novel 2,9-disubstituted-6-morpholino purine derivatives assisted by virtual screening and modelling of class I PI3K isoforms 2023
- 2-Aryladenine derivatives as a potent scaffold for A1, A3 and dual A1/A3 adenosine receptor antagonists: Synthesis and structure-activity relationships. Bioorganic & Medicinal Chemistry. 2019
- 6-Carbohydrazonamidepurines: Convenient precursors for 4,8-disubstituted pyrimido[5,4-d]pyrimidines. Synlett. 2014
- General synthetic approach to 2-phenolic adenine derivatives. Synlett. 2012
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documento
- 4,8-Disubstituted pyrimido[5,4-d]pyrimidines as novel apoptotic independent anticancer agents: synthesis and in vitro activity against HCT116 human colon cancer cells 2015
- New pyrimido[5,4-d]pyrimidines with enhanced anticancer activity on colorectal cancer cells: synthesis, SAR study and mechanism of action 2015
- Synthesis of new 9-(4´-RO-phenyl)-6-cyanopurine derivatives 2015
- Synthesis of new pyrimido[5,4-d]pyrimidines derivatives as potential antitubercular agents 2013
- 6-Amidinopurines as convenient precursors to pyrimido[5,4-d]pyrimidines for sar studies on Mycobacterium tuberculosis 2012
- An efficient synthetic approach to 6-triazolopurines 2012
- 6-Cyanopurines: versatile reagents to generate potentially bioactive compounds 2011
- Synthesis of new 6-carboximidamide purines with potential biological activity 2011
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poster de conferência
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teses